Tizpa
Tizpa contains Tizanidine, which is a short-acting, centrally acting skeletal muscle relaxant. It works by blocking nerve impulses (pain sensations) sent to the brain, specifically acting as an agonist at central alpha-2-adrenergic receptor sites to reduce muscle tone.
Dosage by Body Weight
The initial adult dose is typically 2 mg to 4 mg taken orally every 6 to 8 hours as needed. The dose can be gradually increased if necessary, up to a maximum single dose of 8 mg and a maximum daily dose of 36 mg. Titration must be done carefully under a doctor's supervision. Do not discontinue abruptly.
- Body Weight
- Below 5 kg
- Dose
- Not recommended
- Frequency
- N/A
- Tracking Notes
- Safety and efficacy in pediatric patients have not been established.
- Body Weight
- 5-7 kg
- Dose
- Not recommended
- Frequency
- N/A
- Tracking Notes
- Safety and efficacy in pediatric patients have not been established.
- Body Weight
- 8-10 kg
- Dose
- Not recommended
- Frequency
- N/A
- Tracking Notes
- Safety and efficacy in pediatric patients have not been established.
- Body Weight
- 11-15 kg
- Dose
- Not recommended
- Frequency
- N/A
- Tracking Notes
- Safety and efficacy in pediatric patients have not been established.
- Body Weight
- 16-20 kg
- Dose
- Not recommended
- Frequency
- N/A
- Tracking Notes
- Safety and efficacy in pediatric patients have not been established.
| Body Weight | Dose | Frequency | Tracking Notes |
|---|---|---|---|
| Below 5 kg | Not recommended | N/A | Safety and efficacy in pediatric patients have not been established. |
| 5-7 kg | Not recommended | N/A | Safety and efficacy in pediatric patients have not been established. |
| 8-10 kg | Not recommended | N/A | Safety and efficacy in pediatric patients have not been established. |
| 11-15 kg | Not recommended | N/A | Safety and efficacy in pediatric patients have not been established. |
| 16-20 kg | Not recommended | N/A | Safety and efficacy in pediatric patients have not been established. |
Formulation
Purpose
Used to manage muscle spasticity, cramping, and tightness caused by conditions such as multiple sclerosis, spinal cord injury, or chronic back pain.
Generic Name
TizanidineScheduled Drug
Yes. This medicine should be supplied or used only according to applicable prescription and regulatory requirements.